Publications 2021-2025
| 2025 | |
| 312. | “Photoredox-catalyzed cyclopropanation of allenes towards vinyl-cyclopropanes” |
| H. Xi, Y. Zhang, B. Breit, Chem. Sci., 2025, 16, 16813-16818(link) |
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| 311. | “Hydroformylation of Protected Propargylic Alcohols” |
| A. Veith, V. Agabekov, F. Bauer, B. Breit, Synlett, 2025, ASAP (link) |
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| 310. | “Synthesis of Symmetric and P-Stereogenic Self-Assembling Pyridone-Based Phosphorus Ligands” |
| N. Dierenbach, C. Waloch, F. Bauer, W. Seiche, B. Breit, Synthesis, 2025, ASAP (link) |
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| 309. | “Enantioselective Rhodium-Catalyzed Cycloisomerization of 1,5-Bis(allenes) to Access 1,2-cis-Ethynyl- and Vinyl-Substituted Five-Membered (Hetero)Cycles" |
| F. Panahi, M. Samadani, F. Bauer, B. Breit, Angew. Chem., 2025, 137, e202507993; (link)
Angew. Chem. Int. Ed. 2025, 64, e202507993.(link) |
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| 308. | “Synthesis of monodisperse inorganic polyphosphate polyP10 via a photocaging strategy” |
| S. Moser, G. Hans, J. Ma, T. Haas, N. Jork, F. Bauer, B. Breit, H. J. Jessen, Chem. Sci., 2025, 16, 14635-14645 (link) |
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| 307. | “Light-Mediated Photoredox/Cobalt Dual Catalysis for Multisubstituted Enal Synthesis from Alkyne Feedstock” |
| U. Dutta, B. Breit, ACS Catal., 2025, 15, 13, 11389-11397 (link) |
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| 306. | “Structure-Guided Design of a KMT9 Inhibitor Prodrug with Cellular Activity” |
| S. Wang, N. P. F. Barthes, S. Urban, V. I. Hazai, S. O. Klein, T. Pappert, P. Kümmel, N. Heller, J. Bacher, M. Staudt, J. Ruprecht, L. Peng, M. Sum, C. Berlin, D. Sarraf, P. Regenass, R. Warstat, J. Walz, P. Mishra, L. Zhang, O. Einsle, S. Günther, B. Breit, E. Metzger, M. Jung,R. Schüle, J. Med. Chem., 2025, 68, 13295-13320 (link) |
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| 305. | “A novel inhibitor against the bromodomain PfBDP1 of the malaria pathogen Plasmodium falciparum” |
| M. Amann, R. Warstat, K. K. Rechten, P. Theuer, M. Schustereder, S. Clavey, B. Breit, O. Einsle, M. Huegle, M. Petter, S. Guenther, ChemMedChem, 2025, 20, e202500024 (link) |
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| 304. | “Ring A Cleaving Beta-Diketone Hydrolase Is a Key Enzyme of Steroid Degradation in Anaerobic Bacteria” |
| C. Jacoby, L. Peller, J. Wenzler, M. Lutterbeck, W. Seiche, B. Breit, M. Boll, Environmental Microbiology, 2025, 27, e70034 (link) |
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| 303. | “Ambient Pressure Hydroformylation – A Key Step to Meso-Alkyl BODPYs” |
| L. Miller, F. Bauer, B. Breit, Eur. J. Org. Chem., 2025, 28, e202401089. (link) |
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| 2024 | |
| 302. | “O-p-Methoxyphenyl α-Hydroxycarboxylic Acids as Versatile Hydroxyalkylation Agents for Photocatalysis” |
| C. Nopper, A. Veith, F. Himmelsbach, L. Söhner, B. Breit, Chem. Eur. J. 2024, 31, e202403495. (link) |
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| 301. | “Photochemical Asymmetric Palladium-Catalyzed Allylation Reaction: Expeditious Entry to Chiral 1,2-Amino Alcohols and 1,2-Diamines” |
| H. Xie, H. Chen, U. Dutta, Y. Lan, B. Breit, ACS Catal., 2024, 14,e202400037. (link) |
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| 300. | “Rh-Catalyzed Hydroamination of Allenes: Asymmetric N-Allylation of Amino Acids and Peptides” |
| E. Damer, B. Breit, Chemistry Europe, 2024, e202400037. (link) |
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| 299. | “Rhodium-Catalyzed Enantioselective Intramolecular Hydroalkoxylation of Allenes and Application in the Total Synthesis of (R,R,R)-α-Tocopherol” |
| M. Daiger, S. Giofré, D. Berthold, B. Breit, Chem. Eur. J., 2024, 30, e202402010. (link) |
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| 298. | “Nickel-Catalyzed Regioselective Hydrothiolation of Allenes Enabled by Visible-Light Photoredox Catalysis" |
| H. Xie, B. Breit, Org. Lett., 2024, 26, 21, 4438-4442. (link) |
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| 297. | “Metal- and solvent-free domino reaction of 2-isocyanophenol esters to benzoxazines: long-range 1,5-acyl migration on 1,4-diazabutatriene" |
| A. Akbari, H. Khosravi, F. Bauer, F. Rominger, B. Breit, S. Balalaie, Chem. Commun., 2024, 60, 5421-5424. (link) |
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| 296. | “Azobenzene-Integrated NHC Ligands: A Versatile Platform for Visible-Light-Switchable Metal Catalysis" |
| M. Rölz, B. Butschke, B. Breit, J. Am. Chem. Soc., 2024, 146, 19, 13210-13225. (link) |
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| 295. | “A Tandem Hydroformylation-Organocatalyzed Friedel-Crafts Reaction for the Synthesis of Diindolylmethanes" |
| L. Miller, F. Bauer, B. Breit, Chem. Eur. J, 2024, 30, e202400188. (link) |
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| 294. | “Rhodium-Catalyzed Enantioselective Cyclization of 2-Allenylbenzoxazoles" |
| A. Becker, F. Bauer, B. Breit, Org. Lett., 2024, 26, 2451-2455. (link) |
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| 293. | “Rhodium-Catalyzed Asymmetric Macrocyclization towards Crown Ethers Using Hydroamination of Bis(allenes)" |
| F. Panahi, B. Breit, Angew. Chem., 2024, 136, e202317981; (link)
Angew. Chem. Int. Ed. 2024, 63, e202317981.(link) |
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| 292. | “Carbonylation as a Key Step in New Tandem Reactions – A Route to BODPYs" |
| L. Miller, A. Impelmann, F. Bauer, B. Breit, Chem. Eur. J, 2024, 30, e202303752. (link) Highlighted as Cover Feature: Carbonylation as a Key Step in New Tandem Reactions – A Route to BODIPYs (Chem. Eur. J. 9/2024)
L. Miller, A. Impelmann, F. Bauer, B. Breit, Chem. Eur. J, 2024, 30, e202400146. (link)
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| 2023 | |
| 291. | “Rhodium-Catalyzed Allylic Addition as an Atom-Efficient Approach in Total Synthesis" |
| F. Panahi, F. Bauer, B. Breit, Acc. Chem. Res., 2023, 56, 24, 3676–3693. (link) |
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| 290. | “A novel pan-selective bromodomain inhibitor for epigenetic drug design" |
| R. Warstat, M. Pervaiz, P. Regenass, M. Amann, K. Schmidtkunz, O. Einsle, M. Jung, B. Breit, M. Hügle, S. Günther European journal of medicinal chemistry, 2023, 249 , 115139. (link) |
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| 289. | “A Highly Active Hydroformylation Catalyst Using a Self-Assembling Bis-N-Pyrrolyl Phosphine Ligand" |
| F. Bauer, N. Dierenbach, B. Breit Asian J. Org. Chem., 2023, 12 , e2023002. (link) |
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| 288. | “Rhodium-catalyzed diastereoselective synthesis of highly substituted morpholines from nitrogen-tethered allenols" |
| A. Ziyaei Halimehjani, B. Breit Chem. Commun., 2023, 59 , ASAP. (link) |
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| 287. | “Visible-light induced metal-free intramolecular reductive cyclisations of ketones with alkynes and allenes" |
| N. Tang, R. J. Zachmann, H. Xie, J. Zheng, B. Breit Chem. Commun., 2023, 59 , 2122-2125. (link) |
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| 286. | “Acenaphthoimidazolylidene-Ligated Palladacycle Enabled Suzuki–Miyaura Cross-Coupling Employing Equimolar Organoboron for Tri-Ortho-Substituted Bi(hetero)aryls and Teraryls" |
| K. Wang, H. Yang, F. Bauer, B. Breit, W. Fang Chem. Eur. J., 2023, 29 , e2023007. (link) |
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| 285. | “Nickel(0)-Catalyzed Hydrocyanation of Terminal Allenes: A Regio- and Enantioselective Approach to Branched Allylic Nitriles" |
| T. Bury, S. Kullmann, B. Breit, Adv. Synth. Catal., 2023, 365, 335-341. (link) |
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| 284. | “A Diastereoselective Cascade Annulation Approach to Bridged Polycyclic Heterocycles Involving an Unexpected Rearrangement" |
| A. Nikbakht, A. Ebrahimi Valdani, H. Z. Tejeneki, A. Abbasi Kejani, N. S. Alavijeh, F. Bauer, F. Darvish, B. Breit, S. Balalaie, Org. Lett., 2023, 25, 16-20. (link) |
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| 2022 | |
| 283. | “Synthesis of β-Allenylamines by Addition of Chloroprene Grignards to N-Boc Imines" |
| A. G. A. Geissler, B. Breit, Org. Lett., 2022, 24, 7967-7971. (link)
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| 282. | “Rhodium-Catalyzed Dynamic Kinetic Resolution of Racemic Internal Allenes towards Chiral Allylated Triazoles and Tetrazoles" |
| S. V. Sieger, I. Lubins, B. Breit, Catalysts., 2022, 12, 1209. (link)
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| 281. | “Hydrofunctionalization of Propadiene – New Life for a Previously Unwanted Product" |
| S. V. Sieger, I. Lubins, B. Breit, ACS Catal., 2022, 12, 11301-11305. (link)
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| 280. | “Regio- and Diastereoselective Decarboxylative Allylation of N-Aryl α-Amino Acids by Dual Photoredox/Nickel Catalysis" |
| J. Zheng, C. Nopper, R. Bibi, A. Nikbakht, F. Bauer, B. Breit, ACS Catal., 2022, 12, 5949-5960. (link)
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| 279. | “Organophotoredox/Ni-Cocatalyzed Allylation of Allenes: Regio- and Diastereoselective Access to Homoallylic Alcohols" |
| H. Xie, B. Breit, ACS Catal., 2022, 12, 3249-3255. (link)
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| 278. | “Regio-, Diastereo-, and Enantioselective Decarboxylative Hydroaminoalkylation of Dienol Ethers Enabled by Dual Palladium/Photoredox Catalysis" |
| J. Zheng, N. Tang, H. Xie, B. Breit, Angew. Chem., 2022, 134, e202317981; (link)
Angew. Chem. Int. Ed., 2022, 61, e202317981.(link) |
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| 277. | “Rhodium-catalyzed regioselective addition of thioacids to terminal allenes: enantioselective access to branched allylic thioesters" |
| A. Z. Halimehjani, B. Breit, Chem. Commun., 2022, 58, 1704-1707. (link)
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| 276. | “Phosphine Ligands with Acylguanidinium Groups as Substrate-directing Unit" |
| F. Bauer, B. Breit in "Supramolecular Catalysis: New Directions and Developments", (Ed. P. W. N. M. van Leeuwen and M. Raynal), Wiley-VCH, Weinheim 2022, 179-199. (link)
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| 275. | “Supramolecular Construction of Bidentate Ligands Through Self-assembly by Hydrogen Bonding" |
| F. Bauer, B. Breit in "Supramolecular Catalysis: New Directions and Developments", (Ed. P. W. N. M. van Leeuwen and M. Raynal), Wiley-VCH, Weinheim 2022, 1-25. (link)
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| 2021 | |
| 274. | “Synthesis of (−)-(R)-Sitagliptin by RhI-Catalyzed Asymmetric Hydroamination" |
| D. Berthold, B. Breit, Eur. J. Org. Chem., 2021, 6247-6249. (link)
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| 273. | “Synthesis of (−)-(R)-Sitagliptin by RhI-Catalyzed Asymmetric Hydroamination" |
| A. G. A. Geissler, J. R. Riesterer, B. Breit, Org. Lett., 2021, 23, 23, 9168-9172. (link)
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| 272. | “Rhodium-Catalyzed Regio- and Diastereoselective Hydroarylation of Allenes: An Unprecedented Ene Reaction" |
| H. J. Ghazvini, H. Khosravi, S. Mirzaei, S. Balalei, B. Breit, ACS Catal., 2021, 11, 14571-14574. (link)
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| 271. | “4-Acyl Pyrrole Capped HDAC Inhibitors: A New Scaffold for Hybrid Inhibitors of BET Proteins and Histone Deacetylases as Antileukemia Drug Leads" |
| L. Schäfer-Hübner, R. Warstat, H. Ahlert, P. Mishra, F. B. Kraft,, J. Schliehe-Diecks, A. Schöler, A. Borkhardt, B. Breit, S. Bathia, M. Hügle, S. Günther, F. K. Hansen, J. Med. Chem., 2021, 64, 14620-14646. (link)
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| 270. | “Pharmacokinetic study of the novel phosphocholine derivative 3-dibutylaminopropylphosphonic acid by LC-MS couping" |
| M. G. Kather, J. Zeller, D. Plattner, B. Breit, S. Kreuzaler, G. Krippner, K. Peter, S. U. Eisenhardt, B. Kammerer, J. Chromat. B, 2021, 1186, 122998. (link)
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| 269. | “Cobalt-Catalyzed Hydroboration of Terminal and Internal Alkynes" |
| M. J. González, F. Bauer , B. Breit, Org. Lett., 2021, 23, 8199-8203. (link)
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| 268. | “Tandem Photocatalysis Protocol for Hydrogen Generation/Olefin Hydrogenation Using Pd-g-C3N4-Imine/TiO2 Nanoparticles" |
| M. Jafarpour, F. Feizpour, A. Rezaeifard, N. Pourmorteza, B. Breit, Inorg Chem., 2021, 60, 9484-9495. (link)
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| 267. | “Ruthenium-Catalyzed Enantioselective Addition of Carboxylic Acids to Allenes" |
| J.-L. Hu, F. Bauer , B. Breit, ACS Catal., 2021, 11, 12301-12306. (link)
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| 266. | “Cu-Catalyzed C-H Allylation of Benzimidazoles with Allenes” |
| Y. Dong, B. Breit, Org. Lett., 2021, 23, 6765-6769. (link)
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| 265. | “Urea-Substituted Tetramethylcyclopentadienyl Ligands for Supramolecularly Accelerated RhIII-Catalyzed ortho-C−H Olefination of Benzoic Acid Derivatives” |
D. Maurer, B. Breit, Chem. Eur. J., 2021, 27, 2643-2648. (link)
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| 264. | “Metabolic reprogramming of inner ear cell line HEI-OC1 after dexamethasone application” |
| M. Kather, S. Koitzsch, B. Breit, S. Plontke, B. Kammerer, A. Liebau, Metabolomics, 2021, https://doi.org/10.1007/s11306-021-01799-y. (link)
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| 263. | “Structure-Based Design, Docking and Binding Free Energy Calculations of A366 Derivatives as Spindlin1 Inhibitors” |
C. Luise, D. Robaa, P. Regenass, D. Maurer, D. Ostrovskyi, L. Seifert, J. Bacher, T. Burgahn, T. Wagner, J. Seitz, H. Greschik, K. Park, Y. Xiong, J. Jin, R. Schüle, B. Breit, M. Jung, W. Sippl, Int. J. Mol. Sci., 2021, 22, 5910. (link)
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| 262. | “Asymmetric hydroalkylation of alkynes and allenes with imidazolidinone derivatives: α-alkenylation of α-amino acids” |
F. Panahi, H. Khosravi, F. Bauer, B. Breit, Chem. Sci., 2021, 12, 7388-7392. (link)
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| 261. | “Rhodium-Catalyzed Stereoselective Cyclization of 3-Allenylindoles and N-Allenyltryptamines to Functionalized Vinylic Spiroindolenines” |
| A. Becker, C. P. Grugel, B. Breit, Org. Lett., 2021, 23, 3788-3792. (link)
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| 260. | “Copper-Catalyzed Cycloisomerization of Unactivated Allene-Tethered O-Propargyl Oximes: A Domino Reaction Sequence toward the Synthesis of Hexahydropayrrolo[3,4-b]azepin-5(4H)-ones” |
A. Nikbakht, K. Amiri, H. Khosravi, Y. Zhou, S. Balalei, B. Breit, Org. Lett., 2021, 23, 3343-3348. (link)
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| 259. | “Addition of Chloroprene Grignards to Aromatic Aldehydes: Synthesis of Homoallenyl Alcohols” |
A. G. A. Geissler, B. Breit, Org. Lett., 2021, 23, 2621-2625. (link)
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| 258. | “Dual Palladium/Photoredox-Catalyzed Enantioselective and Regioselective Decarboxylative Hydroaminoalkylation of Allenes” |
J. Zheng, A. Nikbakht, B. Breit, ACS Catal. 2021, 11, 3343-3350. (link)
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| 257. | “Total Syntheses of Cylindrocyclophanes Exemplifying the Power of Transition-Metal Catalysis in Natural-Product Synthesis” |
D. Berthold, B. Breit, Synlett, 2021, 32, 436-446. (link)
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| 256. | “Metal-Free Domino Oligozyclization Reactions of Enynals and Enyones with Molecular Oxygen” |
A. A. Kejani, H. Khosravi, F. Rominger, S. Balalaie, B. Breit, Org. Lett., 2021, 23, 1291-1295. (link)
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| 255. | “Catalyst Deactivation During Rhodium Complex-Catalyzed Propargylic C−H Activation” |
| S. Möller, N. Jannsen, J. Rüger, H.-J. Drexler, M. Horstmann, F. Bauer, B. Breit, D. Heller, Chem. Eur. J., 2021, 27, 14034-14041. (link)
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